Kisspeptin

Source / Derivation:

Kisspeptin is a naturally occurring peptide derived from the KISS1 gene, originally identified for its role in regulating reproductive hormone signaling. Synthetic analogs are developed to target the hypothalamic–pituitary–gonadal (HPG) axis with high specificity and bioactivity.

Kisspeptin

Mechanism of Action:

Kisspeptin binds to GPR54 (KISS1R) receptors in the hypothalamus, stimulating the release of gonadotropin-releasing hormone (GnRH). This, in turn, increases luteinizing hormone (LH) and follicle-stimulating hormone (FSH) secretion, supporting downstream sex steroid production and reproductive endocrine function.

Clinical Relevance & Potential Outcomes:

Research suggests Kisspeptin may support enhanced reproductive hormone regulation, improved fertility parameters, and modulation of endocrine balance. It has potential applications in reproductive endocrinology, delayed puberty, and hormone-related therapeutic interventions.

Intended Clinical Application:

Kisspeptin may be relevant for patients requiring support for reproductive hormone optimization, fertility management, or restoration of HPG axis function.

Formulation & Quality Specifications:

Delivered as a liquid prefilled pen
Purity: >98% (HPLC-validated)
Storage: 2–8 °C (refrigerated)
Documentation: Full CoA and MSDS available

Concentration:

Frequency:

Dosage (pen clicks):

Duration:

Notes:

5 mg/ml, total 3 ml, total 15 mg

Daily

1 month

A peptide involved in reproductive health, regulating gonadotropin secretion, and supporting fertility and hormonal balance.

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